MedKoo Biosciences, Inc.
Tel:   +1-919-636-5577    Fax:   +1-919-980-4831    Email:   sales@medkoo.com
Search
Login Register
Search
MedKoo Cat#: 524964 | Name: Diltiazem malate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Diltiazem malate is an ACE inhibitor and a non-dihydropyridine calcium channel blocker. It is used in the treatment of hypertension.

Chemical Structure

Diltiazem malate
CAS#144604-00-2 (malate)

Theoretical Analysis

MedKoo Cat#: 524964

Name: Diltiazem malate

CAS#: 144604-00-2 (malate)

Chemical Formula: C26H32N2O9S

Exact Mass: 0.0000

Molecular Weight: 548.61

Elemental Analysis: C, 56.92; H, 5.88; N, 5.11; O, 26.25; S, 5.84

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
42399-41-7 (free base) 144604-00-2 (malate) 33286-22-5 (HCl) 139492-78-7 (maleate)
Synonym
Diltiazem malate; Diltiazem malate; MK-793; Tiamate; UNII-14Y6444DRP.
IUPAC/Chemical Name
(2S,3S)-5-(2-(dimethylamino)ethyl)-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-yl acetate (S)-2-hydroxysuccinate
InChi Key
IUSFTUWHKCSCDY-QTKZZPNDSA-N
InChi Code
InChI=1S/C22H26N2O4S.C4H6O5/c1-15(25)28-20-21(16-9-11-17(27-4)12-10-16)29-19-8-6-5-7-18(19)24(22(20)26)14-13-23(2)3;5-2(4(8)9)1-3(6)7/h5-12,20-21H,13-14H2,1-4H3;2,5H,1H2,(H,6,7)(H,8,9)/t20-,21+;2-/m10/s1
SMILES Code
O=C1[C@H](OC(C)=O)[C@H](C2=CC=C(OC)C=C2)SC3=CC=CC=C3N1CCN(C)C.O=C(O)[C@@H](O)CC(O)=O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 548.61 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Bloomgarden ZT. American Diabetes Association annual meeting, 1997, and the Teczem Consultant Meeting. Diabetic nephropathy. Diabetes Care. 1998 Feb;21(2):315-9. PubMed PMID: 9540001.

View History

Diketone-PEG11-PFP ester

Diketone-PEG11-PFP ester