GI-530159, GI530159, GI 530159, a novel, selective, mechano-sensitive K2P channel opener. Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels.
MedKoo Cat#: 471020
Name: GI-530159
CAS#: 69563-88-8 (free base)
Chemical Formula: C27H20F6N2O2
Exact Mass: 518.1429
Molecular Weight: 518.46
Elemental Analysis: C, 62.55; H, 3.89; F, 21.99; N, 5.40; O, 6.17
Solvent | mg/mL | mM | |
---|---|---|---|
Solubility | |||
DMSO | 51.8 | 100.00 |
The following data is based on the product molecular weight 518.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |