LY 190388 | CAS#105496-35-3 | mu receptor agonist

MedKoo Cat#: 525504 | Name: LY 190388

Description:

WARNING: This product is for research use only, not for human or veterinary use.

LY 190388 is a penicillamine-containing enkephalin analog. It is an mu receptor agonist that produces analgesia..

Chemical Structure

LY 190388

CAS#105496-35-3

Theoretical Analysis

MedKoo Cat#: 525504

Name: LY 190388

CAS#: 105496-35-3

Chemical Formula: C30H41N5O7S

Exact Mass: 615.2727

Molecular Weight: 615.74

Elemental Analysis: C, 58.52; H, 6.71; N, 11.37; O, 18.19; S, 5.21

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

No Data

Synonym

LY 190388; LY190388; LY-190388.

IUPAC/Chemical Name

D-Valine, N-(N-(N-(3-mercapto-N-L-tyrosyl-D-valyl)glycyl)-L-phenylalanyl)-

InChi Key

PMSAWKRESCKOJT-HFOXQMJASA-N

InChi Code

InChI=1S/C30H41N5O7S/c1-17(2)24(29(41)42)34-27(39)22(15-18-8-6-5-7-9-18)33-23(37)16-32-28(40)25(30(3,4)43)35-26(38)21(31)14-19-10-12-20(36)13-11-19/h5-13,17,21-22,24-25,36,43H,14-16,31H2,1-4H3,(H,32,40)(H,33,37)(H,34,39)(H,35,38)(H,41,42)/t21-,22-,24+,25-/m0/s1

SMILES Code

CC(C)[C@H](C(O)=O)NC([C@H](CC1=CC=CC=C1)NC(CNC([C@@H](C(C)(S)C)NC([C@H](CC2=CC=C(C=C2)O)N)=O)=O)=O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 615.74 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Leander JD, Gesellchen PD, Mendelsohn LG. Comparison of two penicillamine-containing enkephalins: mu, not delta, activity produces analgesia. Neuropeptides. 1986 Aug-Sep;8(2):119-25. PubMed PMID: 3020472.