Basimglurant is a potent, selective, and safe mGlu5 inhibitor with good oral bioavailability and long half-life supportive of once-daily administration, good brain penetration, and high in vivo potency.
MedKoo Cat#: 126417
Name: Basimglurant sulfate
CAS#: 1034442-21-1 (sulfate)
Chemical Formula: C18H15ClFN3O4S
Exact Mass: 423.0456
Molecular Weight: 423.84
Elemental Analysis: C, 51.01; H, 3.57; Cl, 8.36; F, 4.48; N, 9.91; O, 15.10; S, 7.56
The following data is based on the product molecular weight 423.84 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
