CAY10771 is a dual agonist of farnesoid X receptor (FXR) and peroxisome proliferator-activated receptor δ (PPARδ). It activates FXR and PPARδ in reporter assays using HEK293T cells and is selective for these receptors over retinoic acid receptor α (RARα), retinoid X receptor α (RXRα), PPARα, PPARγ, and liver X receptor α (LXRα) at 10 µM.
MedKoo Cat#: 463929
Name: CAY10771
CAS#: 2522599-79-5
Chemical Formula: C28H25Cl3N2O4
Exact Mass: 558.0880
Molecular Weight: 559.87
Elemental Analysis: C, 60.07; H, 4.50; Cl, 19.00; N, 5.00; O, 11.43
The following data is based on the product molecular weight 559.87 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
