Bromopride HCl | CAS# 52423-56-0 (HCl) | dopamine D2 receptor blocker

MedKoo Cat#: 412426 | Name: Bromopride HCl

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Bromopride HCl is the salt form of Bromopride, a dopamine D2 receptor blocker. Bromopride exerts is a gastrointestinal prokinetic exploited clinically for the management of motor disorders of the upper gastrointestinal tract, including functional dyspepsia, gastric stasis of various origins and emesis.

Chemical Structure

Bromopride HCl

CAS#52423-56-0 (HCl)

Theoretical Analysis

MedKoo Cat#: 412426

Name: Bromopride HCl

CAS#: 52423-56-0 (HCl)

Chemical Formula: C14H23BrClN3O2

Exact Mass: 0.0000

Molecular Weight: 380.71

Elemental Analysis: C, 44.17; H, 6.09; Br, 20.99; Cl, 9.31; N, 11.04; O, 8.40

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

4093-35-0 (free base) 52423-56-0 (HCl)

Synonym

Bromopride hydrochloride; Cascapride; Opridan; Viaben; Bromopride HCl

IUPAC/Chemical Name

4-Amino-5-bromo-N-(2-(diethylamino)ethyl)-2-methoxybenzamide monohydrochloride

InChi Key

SGQFXUUDHWNAIN-UHFFFAOYSA-N

InChi Code

InChI=1S/C14H22BrN3O2.ClH/c1-4-18(5-2)7-6-17-14(19)10-8-11(15)12(16)9-13(10)20-3;/h8-9H,4-7,16H2,1-3H3,(H,17,19);1H

SMILES Code

O=C(NCCN(CC)CC)C1=CC(Br)=C(N)C=C1OC.[H]Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 380.71 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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