MedKoo Cat#: 462199 | Name: SA57

Description:

WARNING: This product is for research use only, not for human or veterinary use.

SA57 is a potent, selective FAAH inhibitor.

Chemical Structure

SA57
SA57
CAS#1346169-63-8

Theoretical Analysis

MedKoo Cat#: 462199

Name: SA57

CAS#: 1346169-63-8

Chemical Formula: C17H23ClN2O3

Exact Mass: 338.1397

Molecular Weight: 338.83

Elemental Analysis: C, 60.26; H, 6.84; Cl, 10.46; N, 8.27; O, 14.17

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
SA57
IUPAC/Chemical Name
2-(methylamino)-2-oxoethyl 4-(4-chlorophenethyl)piperidine-1-carboxylate
InChi Key
JFSSVCSHPDLFCM-UHFFFAOYSA-N
InChi Code
InChI=1S/C17H23ClN2O3/c1-19-16(21)12-23-17(22)20-10-8-14(9-11-20)3-2-13-4-6-15(18)7-5-13/h4-7,14H,2-3,8-12H2,1H3,(H,19,21)
SMILES Code
ClC1=CC=C(CCC2CCN(C(OCC(NC)=O)=O)CC2)C=C1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 338.83 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Niphakis MJ, Johnson DS, Ballard TE, Stiff C, Cravatt BF. O-hydroxyacetamide carbamates as a highly potent and selective class of endocannabinoid hydrolase inhibitors. ACS Chem Neurosci. 2012;3(5):418-426. doi:10.1021/cn200089j 2: Owens RA, Ignatowska-Jankowska B, Mustafa M, et al. Discriminative Stimulus Properties of the Endocannabinoid Catabolic Enzyme Inhibitor SA-57 in Mice. J Pharmacol Exp Ther. 2016;358(2):306-314. doi:10.1124/jpet.115.229492