MedKoo Cat#: 573354 | Name: AY 28925

Description:

WARNING: This product is for research use only, not for human or veterinary use.

AY 28925 is a drug which has adrenoceptor activity as well as nonselective beta-adrenoceptor intrinsic efficacy. AY 28925 has been shown to relax tracheal smooth muscle in guinea pigs.

Chemical Structure

AY 28925
AY 28925
CAS#101565-18-8

Theoretical Analysis

MedKoo Cat#: 573354

Name: AY 28925

CAS#: 101565-18-8

Chemical Formula: C21H25N3O2

Exact Mass: 351.1947

Molecular Weight: 351.45

Elemental Analysis: C, 71.77; H, 7.17; N, 11.96; O, 9.10

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
No Data
Synonym
AY 28925
IUPAC/Chemical Name
1H-Indole-7-carboxamide, 5-(1-hydroxy-2-((1-methyl-3-phenylpropyl)amino)ethyl)-
InChi Key
DEXHZSZLIVQAPC-UHFFFAOYSA-N
InChi Code
1S/C21H25N3O2/c1-14(7-8-15-5-3-2-4-6-15)24-13-19(25)17-11-16-9-10-23-20(16)18(12-17)21(22)26/h2-6,9-12,14,19,23-25H,7-8,13H2,1H3,(H2,22,26)
SMILES Code
c1c(cc2cc[nH]c2c1C(N)=O)[C@@H](CN[C@@H](CCc1ccccc1)C)O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 351.45 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Heaslip RJ, Giesa FR, Rimele TJ, Grimes D. Demonstration of the beta 2-adrenoceptor intrinsic efficacy of AY-28,925 using the PGF2 alpha-contracted guinea-pig trachea. Eur J Pharmacol. 1987 Jun 4;137(2-3):179-84. PubMed PMID: 2886349. 2: Rimele TJ, Heaslip RJ, Lee DK, Grimes D. In vitro characterization of the adrenoceptor activity of AY-28,925. J Pharmacol Exp Ther. 1986 Oct;239(1):1-8. PubMed PMID: 2876089.