Gabazine hydrobromide | CAS#104104-50-9 | GABAA receptor antagonist

MedKoo Cat#: 527770 | Name: Gabazine hydrobromide

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Gabazine is a specific GABAA receptor antagonist.

Chemical Structure

Gabazine hydrobromide

CAS#104104-50-9 (HBr)

Theoretical Analysis

MedKoo Cat#: 527770

Name: Gabazine hydrobromide

CAS#: 104104-50-9 (HBr)

Chemical Formula: C15H18BrN3O3

Exact Mass: 0.0000

Molecular Weight: 368.23

Elemental Analysis: C, 48.93; H, 4.93; Br, 21.70; N, 11.41; O, 13.03

Price and Availability

Size	Price	Availability	Quantity
10mg	USD 350.00	2 Weeks
50mg	USD 850.00	2 Weeks

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Related CAS #

105538-73-6 (free base) 104104-50-9 (HBr)

Synonym

Gabazine hydrobromide; Gabazine HBr; SR95531; SR 95531; SR-95531

IUPAC/Chemical Name

6-imino-3-(4-methoxyphenyl)-1(6H)-pyridazinebutanoic acid, monohydrobromide

InChi Key

GFZHNFOGCMEYTA-UHFFFAOYSA-N

InChi Code

InChI=1S/C15H17N3O3.BrH/c1-21-12-6-4-11(5-7-12)13-8-9-14(16)18(17-13)10-2-3-15(19)20;/h4-9,16H,2-3,10H2,1H3,(H,19,20);1H

SMILES Code

N=C1N(CCCC(O)=O)N=C(C2=CC=C(OC)C=C2)C=C1.Br

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 368.23 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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