Btg 502 | CAS#99083-11-1 | insecticide

MedKoo Cat#: 584285 | Name: Btg 502

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Btg 502 activates sodium channel & inhibits batrachotoxinin A-20-alpha-benzoate binding.

Chemical Structure

Btg 502

CAS#99083-11-1

Theoretical Analysis

MedKoo Cat#: 584285

Name: Btg 502

CAS#: 99083-11-1

Chemical Formula: C21H24BrNO

Exact Mass: 385.1041

Molecular Weight: 386.33

Elemental Analysis: C, 65.29; H, 6.26; Br, 20.68; N, 3.63; O, 4.14

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

No Data

Synonym

Btg 502; Btg-502; Btg502

IUPAC/Chemical Name

2,4-Hexadienamide, 6-(5-bromo-2-naphthalenyl)-N-(1,2-dimethylpropyl)-, (E,E)-

InChi Key

FVMPXCCSVGCCRV-LJIKRCSCSA-N

InChi Code

InChI=1S/C21H24BrNO/c1-15(2)16(3)23-21(24)11-6-4-5-8-17-12-13-19-18(14-17)9-7-10-20(19)22/h4-7,9-16H,8H2,1-3H3,(H,23,24)/b5-4+,11-6+

SMILES Code

O=C(NC(C)C(C)C)/C=C/C=C/CC1=CC=C2C(Br)=CC=CC2=C1

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 386.33 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Du Y, Khambay B, Dong K. An important role of a pyrethroid-sensing residue F1519 in the action of the N-alkylamide insecticide BTG 502 on the cockroach sodium channel. Insect Biochem Mol Biol. 2011 Jul;41(7):446-50. doi: 10.1016/j.ibmb.2011.03.005. Epub 2011 Mar 21. PubMed PMID: 21426938; PubMed Central PMCID: PMC3118982. 2: Du Y, Garden D, Khambay B, Zhorov BS, Dong K. Batrachotoxin, pyrethroids, and BTG 502 share overlapping binding sites on insect sodium channels. Mol Pharmacol. 2011 Sep;80(3):426-33. doi: 10.1124/mol.111.072504. Epub 2011 Jun 16. PubMed PMID: 21680776; PubMed Central PMCID: PMC3164329. 3: Ottea JA, Payne GT, Bloomquist JR, Soderlund DM. Activation of sodium channels and inhibition of [3H]batrachotoxinin A-20-alpha-benzoate binding by an N-alkylamide neurotoxin. Mol Pharmacol. 1989 Aug;36(2):280-4. PubMed PMID: 2549384.