Panadiplon | CAS#124423-84-3

MedKoo Cat#: 528409 | Name: Panadiplon

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Panadiplon (also known as FD-10571, FG-10571, U-78875, and NNC-140571) is a gamma-aminobutyric acid receptor agonist potentially for the treatment of anxiety.

Chemical Structure

Panadiplon

CAS#124423-84-3

Theoretical Analysis

MedKoo Cat#: 528409

Name: Panadiplon

CAS#: 124423-84-3

Chemical Formula: C18H17N5O2

Exact Mass: 335.1382

Molecular Weight: 335.37

Elemental Analysis: C, 64.47; H, 5.11; N, 20.88; O, 9.54

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

Panadiplon; FD-10571; FD 10571; FD10571; FG-10571; FG10571; FG 10571; U-78875; U78875; U 78875; NNC-140571; NNC 140571; NNC140571

IUPAC/Chemical Name

3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-isopropylimidazo[1,5-a]quinoxalin-4(5H)-one

InChi Key

ZGEGOFCLSWVVKG-UHFFFAOYSA-N

InChi Code

InChI=1S/C18H17N5O2/c1-10(2)23-13-6-4-3-5-12(13)22-9-19-14(15(22)18(23)24)16-20-17(25-21-16)11-7-8-11/h3-6,9-11H,7-8H2,1-2H3

SMILES Code

O=C1C2=C(C3=NOC(C4CC4)=N3)N=CN2C5=C(C=CC=C5)N1C(C)C

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Panadiplon pretreatment resulted in leftward shifts in the pentobarbital dose-response function but predominantly rightward shifts of the triazolam dose-response function. During normoxia both cotreatments with panadiplon resulted in significantly higher glycogen levels than in panadiplon cultures alone. These results suggest that cellular glycogen and subsequently ATP levels are reduced during panadiplon exposure, metabolically predisposing hepatocytes to hypoxic injury.

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 335.37 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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