Elzasonan citrate is a selective 5-HT1B and 5-HT1D receptor antagonist for the treatment of depression. By preferentially blocking 5-HT1B and 5-HT1D autoreceptors, Elzasonan is thought to enhance serotonergic innervations originating from the raphe nucleus, thereby improving signaling to limbic regions like the hippocampus and prefrontal cortex and ultimately resulting in antidepressant effects.
MedKoo Cat#: 525002
Name: Elzasonan citrate
CAS#: 361343-20-6 (Citrate)
Chemical Formula: C28H31Cl2N3O8S
Exact Mass: 0.0000
Molecular Weight: 640.53
Elemental Analysis: C, 52.50; H, 4.88; Cl, 11.07; N, 6.56; O, 19.98; S, 5.01
The following data is based on the product molecular weight 640.53 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |