BMS-442606 is a 5-HT1A partial agonist. (S)-Enantiomer has advantage of being cleared more slowly from blood compared to the (R)-enantiomer. (R)-Enantiomer showed higher affinity and selectivity for the 5HT1A receptor compared to the (S)-enantiomer.
MedKoo Cat#: 524477
Name: BMS-442606
CAS#: 477930-31-7
Chemical Formula: C21H31N5O3
Exact Mass: 401.2427
Molecular Weight: 401.51
Elemental Analysis: C, 62.82; H, 7.78; N, 17.44; O, 11.95
The following data is based on the product molecular weight 401.51 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
