Synonym
Cycrimine; Pagitane; Cicrimina; Cycriminum; (+)-cycrimine; Cicrimina
IUPAC/Chemical Name
1-cyclopentyl-1-phenyl-3-piperidin-1-ylpropan-1-ol
InChi Key
SWRUZBWLEWHWRI-UHFFFAOYSA-N
InChi Code
InChI=1S/C19H29NO/c21-19(18-11-5-6-12-18,17-9-3-1-4-10-17)13-16-20-14-7-2-8-15-20/h1,3-4,9-10,18,21H,2,5-8,11-16H2
SMILES Code
C1CCN(CC1)CCC(C2CCCC2)(C3=CC=CC=C3)O
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
Preparing Stock Solutions
The following data is based on the
product
molecular weight
287.44
Batch specific molecular weights may vary
from batch to batch
due to the degree of hydration, which will
affect the solvent
volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass |
1 mg |
5 mg |
10 mg |
| 1 mM |
1.15 mL |
5.76 mL |
11.51 mL |
| 5 mM |
0.23 mL |
1.15 mL |
2.3 mL |
| 10 mM |
0.12 mL |
0.58 mL |
1.15 mL |
| 50 mM |
0.02 mL |
0.12 mL |
0.23 mL |
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2: Sotriffer CA, Liedl KR, Winger RH, Gamper AM, Kroemer RT, Linthicum DS, Rode BM, Varga JM. Heteroligation of a mouse monoclonal IgE antibody (La2) with small molecules, analysed by computer-aided automated docking. Mol Immunol. 1996 Feb;33(2):129-44. PubMed PMID: 8649435.
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7: KAFER JP, POCH GF. [Cycrimine, a new drug in the treatment of Parkinson's disease & Parkinsonism]. Prensa Med Argent. 1957 Apr 5;44(14):1071-5. Spanish. PubMed PMID: 13477721.
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9: NEW AND nonofficial remedies: cycrimine hydrochloride. J Am Med Assoc. 1955 Feb 5;157(6):510-1. PubMed PMID: 13221464.
