Bisulepin is a first-generation antihistamine primarily used for the treatment of allergic conditions such as rhinitis, urticaria, and pruritus. It works by blocking H₁ histamine receptors, thereby reducing the effects of histamine—a chemical involved in allergic reactions. Bisulepin also exhibits sedative and anticholinergic properties due to its ability to cross the blood-brain barrier.
MedKoo Cat#: 146337
Name: Bisulepin
CAS#: 42504-83-6
Chemical Formula: C17H19NS2
Exact Mass: 301.0959
Molecular Weight: 301.47
Elemental Analysis: C, 67.73; H, 6.35; N, 4.65; S, 21.27
The following data is based on the product molecular weight 301.47 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
