GSK205 is an inhibitor of transient receptor potential vanilloid 4 (TRPV4) and transient receptor potential ankyrin 1 (TRPA1; IC50s = 4.19 and 5.56 µM, respectively, for the rat channels).
MedKoo Cat#: 127090
Name: GSK205
CAS#: 1263068-83-2 (HBr)
Chemical Formula: C24H25BrN4S
Exact Mass: 480.0983
Molecular Weight: 481.46
Elemental Analysis: C, 59.87; H, 5.23; Br, 16.60; N, 11.64; S, 6.66
The following data is based on the product molecular weight 481.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
