TUG-2208 is a highly potent GPR84 agonist (EC50= 1.0 nM) with lowered lipophilicity and good to excellent solubility, in vitro permeability, and microsomal stability, which will be valuable tools for exploring the pharmacology and therapeutic prospects of GPR84.
MedKoo Cat#: 126356
Name: TUG-2208
CAS#: N/A
Chemical Formula: C16H12N2O3
Exact Mass: 280.0848
Molecular Weight: 280.28
Elemental Analysis: C, 68.56; H, 4.32; N, 9.99; O, 17.12
The following data is based on the product molecular weight 280.28 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
