Sabcomeline | CAS#159912-53-5 | M1 receptor partial agonist

MedKoo Cat#: 126085 | Name: Sabcomeline

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Sabcomeline, also known as BCI-224; BRL-55473; CEB-2424; SB-202026A, is a selective M1 receptor partial agonist that was under development for the treatment of Alzheimer's disease. It made it to phase III clinical trials before being discontinued due to poor results.

Chemical Structure

Sabcomeline

CAS#159912-53-5 (free base)

Theoretical Analysis

MedKoo Cat#: 126085

Name: Sabcomeline

CAS#: 159912-53-5 (free base)

Chemical Formula: C10H15N3O

Exact Mass: 193.1215

Molecular Weight: 193.25

Elemental Analysis: C, 62.15; H, 7.82; N, 21.74; O, 8.28

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

159912-58-0 (HCl) 159912-53-5(free base)

Synonym

Sabcomeline; SB202026; SB 202026; SB-202026; BCI-224; BRL-55473; CEB-2424; SB-202026A; BCI224; BRL55473; CEB2424; SB202026A

IUPAC/Chemical Name

(R,Z)-N-methoxyquinuclidine-3-carbimidoyl cyanide

InChi Key

IQWCBYSUUOFOMF-QTLFRQQHSA-N

InChi Code

InChI=1S/C10H15N3O/c1-14-12-10(6-11)9-7-13-4-2-8(9)3-5-13/h8-9H,2-5,7H2,1H3/b12-10+/t9-/m0/s1

SMILES Code

[H][C@@]1(CN2CCC1CC2)C(\C#N)=N\OC

Appearance

To be determined

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 193.25 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.