Oxomemazine HCl | CAS# 4784-40-1 | antiallergic agent

MedKoo Cat#: 414689 | Name: Oxomemazine HCl

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Oxomemazine is an antihistamine and anticholinergic used for the treatment of cough. Oxomemazine is selective for M1 muscarinic receptors. Oxomemazine could be classified as a selective drug for M1 receptors and also demonstrate that rat cerebral microsomes contain three different subtypes of M1, M3 and the other site which is different from M1, M2 and M3 receptors.

Chemical Structure

Oxomemazine HCl

CAS#4784-40-1 (HCl)

Theoretical Analysis

MedKoo Cat#: 414689

Name: Oxomemazine HCl

CAS#: 4784-40-1 (HCl)

Chemical Formula: C18H23ClN2O2S

Exact Mass: 0.0000

Molecular Weight: 366.90

Elemental Analysis: C, 58.92; H, 6.32; Cl, 9.66; N, 7.64; O, 8.72; S, 8.74

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

3689-50-7 (free base) 4784-40-1 (HCl)

Synonym

Oxomemazine hydrochloride; Oxomemazine HCl

IUPAC/Chemical Name

N,N,beta-Trimethyl-10H-phenothiazine-10-propylamine 5,5-dioxide monohydrochloride

InChi Key

NPMMOYKGIWLASW-UHFFFAOYSA-N

InChi Code

InChI=1S/C18H22N2O2S.ClH/c1-14(12-19(2)3)13-20-15-8-4-6-10-17(15)23(21,22)18-11-7-5-9-16(18)20;/h4-11,14H,12-13H2,1-3H3;1H

SMILES Code

CC(CN1c2c(S(=O)(c3c1cccc3)=O)cccc2)CN(C)C.Cl

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 366.90 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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