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MedKoo Cat#: 412760 | Name: Serazapine hydrochloride

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Serazapine hydrochloride is an Anti-Anxiety Agent

Chemical Structure

Serazapine hydrochloride
CAS#117581-05-2 (HCl)

Theoretical Analysis

MedKoo Cat#: 412760

Name: Serazapine hydrochloride

CAS#: 117581-05-2 (HCl)

Chemical Formula: C22H24ClN3O2

Exact Mass: 397.1557

Molecular Weight: 0.00

Elemental Analysis: C, 66.41; H, 6.08; Cl, 8.91; N, 10.56; O, 8.04

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
117581-05-2 (HCl) 115313-22-9 (free base)
Synonym
Serazapine hydrochloride; CGS15040A; CGS-15040A; CGS 15040A
IUPAC/Chemical Name
2H,10H-Indolo(2,1-c)pyrazino(1,2-a)(1,4)benzodiazepine-16-carboxylic acid, 1,3,4,16b-tetrahydro-2-methyl-, methyl ester, monohydrochloride
InChi Key
YEITZTKANLXOTH-UHFFFAOYSA-N
InChi Code
InChI=1S/C22H23N3O2.ClH/c1-23-11-12-24-17-9-5-3-7-15(17)13-25-18-10-6-4-8-16(18)20(22(26)27-2)21(25)19(24)14-23;/h3-10,19H,11-14H2,1-2H3;1H
SMILES Code
O=C(C1=C2C(CN(C)CC3)N3C4=CC=CC=C4CN2C5=C1C=CC=C5)OC.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 0.00 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Luders RC, Brunner LA, Shum LY, Ross HD, Das H. Determination of CGS 15040A in human plasma by liquid chromatography. J Pharm Biomed Anal. 1991;9(4):351-5. doi: 10.1016/0731-7085(91)80205-n. PMID: 1680469. 2: Katz RJ, Landau PS, Lott M, Bystritsky A, Diamond B, Hoehn-Saric R, Rosenthal M, Weise C. Serotonergic (5-HT2) mediation of anxiety-therapeutic effects of serazepine in generalized anxiety disorder. Biol Psychiatry. 1993 Jul 1-15;34(1-2):41-4. doi: 10.1016/0006-3223(93)90254-b. PMID: 8104044.