MedKoo Cat#: 463576 | Name: SR10658

Description:

WARNING: This product is for research use only, not for human or veterinary use.

SR10658 is a NR4A Ligand (full-length Nurr1 EC50 = 4.1nM). The NR4A nuclear receptor transcription factors regulate important physiological processes including cellular homeostasis, metabolic regulation, apoptosis, and cell differentiation.

Chemical Structure

SR10658
SR10658
CAS#unknown

Theoretical Analysis

MedKoo Cat#: 463576

Name: SR10658

CAS#: unknown

Chemical Formula: C20H18N2O3

Exact Mass: 334.1317

Molecular Weight: 334.38

Elemental Analysis: C, 71.84; H, 5.43; N, 8.38; O, 14.35

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
SR10658; SR 10658; SR-10658;
IUPAC/Chemical Name
6-(4-methoxyphenyl)-5-methyl-3-phenyl-5,7a-dihydroisoxazolo[4,5-c]pyridin-4(3aH)-one
InChi Key
FVPMPUUOFPPKQC-UHFFFAOYSA-N
InChi Code
InChI=1S/C20H18N2O3/c1-22-16(13-8-10-15(24-2)11-9-13)12-17-18(20(22)23)19(21-25-17)14-6-4-3-5-7-14/h3-12,17-18H,1-2H3
SMILES Code
O=C(N1C)C2C(ON=C2C3=CC=CC=C3)C=C1C4=CC=C(OC)C=C4
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 334.38 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL