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MedKoo Cat#: 412659 | Name: CGP 54062

Description:

WARNING: This product is for research use only, not for human or veterinary use.

CGP 54062 is a GABA-B receptor antagonist; CGP 55845 is the (1S,2S)-isomer.

Chemical Structure

CGP 54062
CGP 54062
CAS#148056-42-2

Theoretical Analysis

MedKoo Cat#: 412659

Name: CGP 54062

CAS#: 148056-42-2

Chemical Formula: C18H22Cl2NO2P

Exact Mass: 385.0765

Molecular Weight: 386.25

Elemental Analysis: C, 55.97; H, 5.74; Cl, 18.36; N, 3.63; O, 8.28; P, 8.02

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
CGP 54062; CGP54062; CGP-54062
IUPAC/Chemical Name
Phosphinic acid, (3-((1-(3,4-dichlorophenyl)ethyl)amino)-2-hydroxpropyl)(phenylmethyl)-
InChi Key
RPVSIAKLYXUQLS-UHFFFAOYSA-N
InChi Code
InChI=1S/C18H22Cl2NO2P/c1-14(16-8-9-17(19)18(20)12-16)21-10-5-11-24(22,23)13-15-6-3-2-4-7-15/h2-4,6-9,12,14,21H,5,10-11,13H2,1H3,(H,22,23)
SMILES Code
O=P(CC1=CC=CC=C1)(CCCNC(C2=CC=C(Cl)C(Cl)=C2)C)O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 386.25 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Olpe HR, Steinmann MW, Ferrat T, Pozza MF, Greiner K, Brugger F, Froestl W, Mickel SJ, Bittiger H. The actions of orally active GABAB receptor antagonists on GABAergic transmission in vivo and in vitro. Eur J Pharmacol. 1993 Mar 23;233(2-3):179-86. doi: 10.1016/0014-2999(93)90048-m. PMID: 8385620. 2: Brugger F, Wicki U, Olpe HR, Froestl W, Mickel S. The action of new potent GABAB receptor antagonists in the hemisected spinal cord preparation of the rat. Eur J Pharmacol. 1993 Apr 22;235(1):153-5. doi: 10.1016/0014-2999(93)90836-7. PMID: 8390938.

View History

CGP 47656

CGP 47656

CL 286527

CL 286527

MK-7128

MK-7128