MedKoo Cat#: 513674 | Name: CGP 47656

Description:

WARNING: This product is for research use only, not for human or veterinary use.

CGP 47656 is GABAB receptor agonist.

Chemical Structure

CGP 47656
CGP 47656
CAS#133345-73-0

Theoretical Analysis

MedKoo Cat#: 513674

Name: CGP 47656

CAS#: 133345-73-0

Chemical Formula: C4H10F2NO2P

Exact Mass: 173.0417

Molecular Weight: 173.10

Elemental Analysis: C, 27.76; H, 5.82; F, 21.95; N, 8.09; O, 18.49; P, 17.89

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
CGP 47656; CGP47656; CGP-47656.
IUPAC/Chemical Name
3-aminopropyl-(difluoromethyl)phosphinic acid
InChi Key
TXAHGWWWANKBDA-UHFFFAOYSA-N
InChi Code
InChI=1S/C4H10F2NO2P/c5-4(6)10(8,9)3-1-2-7/h4H,1-3,7H2,(H,8,9)
SMILES Code
O=P(C(F)F)(CCCN)O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 173.10 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Marcoli M, Scarrone S, Maura G, Bonanno G, Raiteri M. A subtype of the gamma-aminobutyric acid(B) receptor regulates cholinergic twitch response in the guinea pig ileum. J Pharmacol Exp Ther. 2000 Apr;293(1):42-7. PubMed PMID: 10734151. 2: Raiteri M, Bonanno G, Paudice P, Cavazzani P, Schmid G. Human brain cholecystokinin: release of cholecystokinin-like immunoreactivity (CCK-LI) from isolated cortical nerve endings and its modulation through GABA(B) receptors. J Pharmacol Exp Ther. 1996 Aug;278(2):747-51. PubMed PMID: 8768727. 3: Bonanno G, Gemignani A, Schmid G, Severi P, Cavazzani P, Raiteri M. Human brain somatostatin release from isolated cortical nerve endings and its modulation through GABAB receptors. Br J Pharmacol. 1996 Jul;118(6):1441-6. PubMed PMID: 8832070; PubMed Central PMCID: PMC1909667. 4: Gemignani A, Paudice P, Bonanno G, Raiteri M. Pharmacological discrimination between gamma-aminobutyric acid type B receptors regulating cholecystokinin and somatostatin release from rat neocortex synaptosomes. Mol Pharmacol. 1994 Sep;46(3):558-62. PubMed PMID: 7935338.