Estradiol sulfamate is a steroid sulfatase (STS) inhibitor which is under development for the treatment of endometriosis. It is the C3 sulfamate ester of estradiol, and was originally thought to be a prodrug of estradiol.
MedKoo Cat#: 463291
Name: Estradiol sulfamate
CAS#: 172377-52-5 (sulfamate)
Chemical Formula: C18H25NO4S
Exact Mass: 351.1504
Molecular Weight: 351.46
Elemental Analysis: C, 61.51; H, 7.17; N, 3.99; O, 18.21; S, 9.12
The following data is based on the product molecular weight 351.46 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
