IACS-6274, also known as IPN60090, is a potent, selective and orally active glutaminase inhibitor with potential antineoplastic and immunostimulating activities. IPN60090 selectively targets, binds to and inhibits human glutaminase, an enzyme that is essential for the conversion of the amino acid glutamine into glutamate.
MedKoo Cat#: 207123
Name: IACS-6274 HCl
CAS#: 2102101-72-2 (HCl)
Chemical Formula: C24H29Cl2F3N8O3
Exact Mass: 532.2158
Molecular Weight: 605.44
Elemental Analysis: C, 47.61; H, 4.83; Cl, 11.71; F, 9.41; N, 18.51; O, 7.93
The following data is based on the product molecular weight 605.44 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
