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MedKoo Cat#: 585213 | Name: Endixaprine

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Endixaprine is an anticonvulsant.

Chemical Structure

Endixaprine
Endixaprine
CAS#93181-85-2

Theoretical Analysis

MedKoo Cat#: 585213

Name: Endixaprine

CAS#: 93181-85-2

Chemical Formula: C15H15Cl2N3O

Exact Mass: 323.0592

Molecular Weight: 324.21

Elemental Analysis: C, 55.57; H, 4.66; Cl, 21.87; N, 12.96; O, 4.93

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Endixaprine; SR-41378; SR41378; SR 41378
IUPAC/Chemical Name
4-Piperidinol, 1-(6-(2,4-dichlorophenyl)-3-pyridazinyl)-
InChi Key
COWWILCLLRVLSC-UHFFFAOYSA-N
InChi Code
InChI=1S/C15H15Cl2N3O/c16-10-1-2-12(13(17)9-10)14-3-4-15(19-18-14)20-7-5-11(21)6-8-20/h1-4,9,11,21H,5-8H2
SMILES Code
OC1CCN(C2=NN=C(C3=CC=C(Cl)C=C3Cl)C=C2)CC1
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 324.21 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Stanková L, Mares P. Antimetrazol action of two potential anticonvulsants, CM 40907 and SR 41378, in immature rats. Physiol Res. 1992;41(6):451-7. PubMed PMID: 1299328. 2: Santucci V, Rocher D, Veyrun J, Bizière K. Quantitative electroencephalographic profile of 3-(4-hydroxy-1-piperidinyl)-6-(2,4-dichlorophenyl)-pyridazine (SR 41378) in the rat. Naunyn Schmiedebergs Arch Pharmacol. 1986 Jun;333(2):186-9. PubMed PMID: 2875399. 3: Perio A, Chambon JP, Calassi R, Heaulme M, Biziere K. Evaluation of two anticonvulsant amino-pyridazine derivatives in the conflict test in rats. J Pharmacol Exp Ther. 1986 Nov;239(2):542-7. PubMed PMID: 3095540.

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