SR-12062 is a full agonists of the neurotensin receptor 1 (NTSR1). SR-12062 have an EC50 of 2 μM at NTSR1 with full agonist behaviour (Emax=100%), showing a higher efficacy and ∼90-fold potency improvement compared to parent compound 1 (EC50=178 μM; Emax=17%).
MedKoo Cat#: 555602
Name: SR-12062
CAS#: 1623019-77-1
Chemical Formula: C25H25N3O3
Exact Mass: 415.1896
Molecular Weight: 415.49
Elemental Analysis: C, 72.27; H, 6.07; N, 10.11; O, 11.55
The following data is based on the product molecular weight 415.49 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
