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MedKoo Cat#: 573789 | Name: Amlodipine maleate
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Amlodipine maleate is a long-acting dihydropyridine calcium channel blocker effective in the treatment of angina pectoris and hypertension.

Chemical Structure

Amlodipine maleate
Amlodipine maleate
CAS#88150-47-4 (maleate)

Theoretical Analysis

MedKoo Cat#: 573789

Name: Amlodipine maleate

CAS#: 88150-47-4 (maleate)

Chemical Formula: C24H29ClN2O9

Exact Mass: 524.1562

Molecular Weight: 524.95

Elemental Analysis: C, 54.91; H, 5.57; Cl, 6.75; N, 5.34; O, 27.43

Price and Availability

Size Price Availability Quantity
250mg USD 250.00 2 Weeks
500mg USD 400.00 2 Weeks
1g USD 650.00 2 Weeks
2g USD 1,050.00 2 Weeks
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Related CAS #
246852-12-0 (mesylate) 440358-84-9 (mesylate hydrate) 88150-47-4 (maleate)
Synonym
Amlodipine (+-)-form maleate, Amlodipine maleate, Amvaz
IUPAC/Chemical Name
3,5-Pyridinedicarboxylic acid, 2-((2-aminoethoxy)methyl)-4-(2-chlorophenyl)-1,4-dihydro-6-methyl-, 3-ethyl 5-methyl ester, (+-)-, (Z)-2-butenedioate (1:1)
InChi Key
TZNOWAJJWCGILX-BTJKTKAUSA-N
InChi Code
1S/C20H25ClN2O5.C4H4O4/c1-4-28-20(25)18-15(11-27-10-9-22)23-12(2)16(19(24)26-3)17(18)13-7-5-6-8-14(13)21;5-3(6)1-2-4(7)8/h5-8,17,23H,4,9-11,22H2,1-3H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
SMILES Code
C=1([C@@H](C(=C(NC1COCCN)C)C(OC)=O)c1c(cccc1)Cl)C(OCC)=O.OC(\C=C/C(O)=O)=O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 524.95 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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