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MedKoo Cat#: 598773 | Name: LG 82-4-00

Description:

WARNING: This product is for research use only, not for human or veterinary use.

LG 82-4-00 is a thromboxane inhibitor.

Chemical Structure

LG 82-4-00
LG 82-4-00
CAS#91505-18-9

Theoretical Analysis

MedKoo Cat#: 598773

Name: LG 82-4-00

CAS#: 91505-18-9

Chemical Formula: C10H11ClN2O3S

Exact Mass:

Molecular Weight: 274.72

Elemental Analysis: C, 43.72; H, 4.04; Cl, 12.90; N, 10.20; O, 17.47; S, 11.67

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
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Synonym
LG 82-4-00; LG-82-4-00; LG82-4-00; LG 82400; LG-82400; LG82400;
IUPAC/Chemical Name
5-(2-(1H-imidazol-1-yl)ethoxy)thiophene-2-carboxylic acid hydrochloride
InChi Key
JBOAEUXWXAMIMH-UHFFFAOYSA-N
InChi Code
InChI=1S/C10H10N2O3S.ClH/c13-10(14)8-1-2-9(16-8)15-6-5-12-4-3-11-7-12;/h1-4,7H,5-6H2,(H,13,14);1H
SMILES Code
O=C(C1=CC=C(OCCN2C=CN=C2)S1)O.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info
Product Data
Product Data
Instruction
View handling instruction
Biological target:
LG 82-4-00 is a thromboxane inhibitor.
In vitro activity:
TBD
In vivo activity:
TBD

Preparing Stock Solutions

The following data is based on the product molecular weight 274.72 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Formulation protocol:
TBD
In vitro protocol:
TBD
In vivo protocol:
TBD
1: Smith EF 3rd, Darius H, Ferber H, Schrör K. Inhibition of thromboxane and 12-HPETE formation by dazoxiben and its two thiophenic acid-substituted derivatives. Eur J Pharmacol. 1985 Jun 7;112(2):161-9. PubMed PMID: 3896821. 2: Asai F, Schrör K. Different effects of thromboxane synthetase inhibition on PGI2 and PGE2 synthesis in human vascular tissue bathed in clotting blood. Prog Clin Biol Res. 1987;242:259-64. PubMed PMID: 3313413.