Levofacetoperane | CAS#24558-01-8 | psychostimulant

MedKoo Cat#: 598724 | Name: Levofacetoperane

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Levofacetoperane is a sympathomimetic central nervous system stimulant and is commonly used to treat depression. Levophacetoperane is also a known analeptic and is strongly linked to apnea reversal in dogs after a single intravenous injection.

Chemical Structure

Levofacetoperane

CAS#24558-01-8 (free base)

Theoretical Analysis

MedKoo Cat#: 598724

Name: Levofacetoperane

CAS#: 24558-01-8 (free base)

Chemical Formula: C14H19NO2

Exact Mass: 233.1416

Molecular Weight: 233.31

Elemental Analysis: C, 72.07; H, 8.21; N, 6.00; O, 13.71

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

24558-01-8 (free base) 23257-56-9 (HCl)

Synonym

Levofacetoperane; Lidepran;

IUPAC/Chemical Name

phenyl(piperidin-2-yl)methyl acetate

InChi Key

BKPLVPRTTWIDNL-UHFFFAOYSA-N

InChi Code

InChI=1S/C14H19NO2/c1-11(16)17-14(12-7-3-2-4-8-12)13-9-5-6-10-15-13/h2-4,7-8,13-15H,5-6,9-10H2,1H3

SMILES Code

CC(OC(C1=CC=CC=C1)C2NCCCC2)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>3 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.03.00

More Info

Product Data

Product Data

Instruction

View handling instruction

Biological target:

Levofacetoperane is a sympathomimetic central nervous system stimulant and is commonly used to treat depression.

In vitro activity:

TBD

In vivo activity:

TBD

Preparing Stock Solutions

The following data is based on the product molecular weight 233.31 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

Formulation protocol:

TBD

In vitro protocol:

TBD

In vivo protocol:

TBD

1: SABBATINI F. [FOREIGN PSYCHOPHARMACOLOGICAL DRUGS: LEVOFACETOPERANE (8228 RP)]. Minerva Med. 1964 Oct 31;55:3473-6. Italian. PubMed PMID: 14231300. 2: BEAUJARD M, REVOL E. [Clinical tests of the activity of RP 8228 (phacetoperane) in an oligophrenic child]. Pediatrie. 1960;15:310-6. French. PubMed PMID: 13797965. 3: Ramirez A, Vial H, Barailler J, Pacheco H. [Effects of levophacetoperane, pemoline, fenozolone, and centrophenoxine on catecholamines and serotonin uptake in various parts of the rat brain]. C R Acad Sci Hebd Seances Acad Sci D. 1978 Jul 3;187(1):53-6. French. PubMed PMID: 29714.