Synonym
Piperophos; Rilof;
IUPAC/Chemical Name
S-(2-(2-methylpiperidin-1-yl)-2-oxoethyl) O,O-dipropyl phosphorodithioate
InChi Key
UNLYSVIDNRIVFJ-UHFFFAOYSA-N
InChi Code
InChI=1S/C14H28NO3PS2/c1-4-10-17-19(20,18-11-5-2)21-12-14(16)15-9-7-6-8-13(15)3/h13H,4-12H2,1-3H3
SMILES Code
CC1CCCCN1C(CSP(OCCC)(OCCC)=S)=O
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
Biological target:
Piperophos is an organophosphate and anti-androgenic compound.
Preparing Stock Solutions
The following data is based on the
product
molecular weight
353.48
Batch specific molecular weights may vary
from batch to batch
due to the degree of hydration, which will
affect the solvent
volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass |
1 mg |
5 mg |
10 mg |
| 1 mM |
1.15 mL |
5.76 mL |
11.51 mL |
| 5 mM |
0.23 mL |
1.15 mL |
2.3 mL |
| 10 mM |
0.12 mL |
0.58 mL |
1.15 mL |
| 50 mM |
0.02 mL |
0.12 mL |
0.23 mL |
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6: Pehar V, Kolić D, Zandona A, Šinko G, Katalinić M, Stepanić V, Kovarik Z. Selected herbicides screened for toxicity and analysed as inhibitors of both cholinesterases. Chem Biol Interact. 2023 Jul 1;379:110506. doi: 10.1016/j.cbi.2023.110506. Epub 2023 May 2. PMID: 37141932.
