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MedKoo Cat#: 563371 | Name: Amiloride HCl anhydrous
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

Amiloride HCl anhydrous is a Na+ channel blocker. It acts by blocking TRPP3, acid sensing- (ASIC) and mechanogated membrane-ion channels, as well as the Na+/H+ exchanger.

Chemical Structure

Amiloride HCl anhydrous
Amiloride HCl anhydrous
CAS#2016-88-8 (HCl anhydrous)

Theoretical Analysis

MedKoo Cat#: 563371

Name: Amiloride HCl anhydrous

CAS#: 2016-88-8 (HCl anhydrous)

Chemical Formula: C6H9Cl2N7O

Exact Mass: 265.0246

Molecular Weight: 266.08

Elemental Analysis: C, 27.08; H, 3.41; Cl, 26.65; N, 36.85; O, 6.01

Price and Availability

Size Price Availability Quantity
1g USD 220.00 2 Weeks
5g USD 470.00 2 Weeks
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Related CAS #
2609-46-3 (free base) 2016-88-8 (HCl anhydrous) 17440-83-4 (HCl hydrate)
Synonym
Amiloride HCl anhydrous; Amiloride HCl anhydrous
IUPAC/Chemical Name
3,5-Diamino-N-(aminoiminomethyl)-6-chloropyrazinecarboxamide hydrochloride
InChi Key
ACHKKGDWZVCSNH-UHFFFAOYSA-N
InChi Code
InChI=1S/C6H8ClN7O.ClH/c7-2-4(9)13-3(8)1(12-2)5(15)14-6(10)11;/h(H4,8,9,13)(H4,10,11,14,15);1H
SMILES Code
ClC1=C(N)N=C(N)C(C(NC(N)=N)=O)=N1.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>3 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.03.00
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 266.08 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
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