GZ4 | CAS#68312-88-9 | Ca2+ current inhibitor

MedKoo Cat#: 563086 | Name: GZ4

Description:

WARNING: This product is for research use only, not for human or veterinary use.

GZ4 is an inhibitor of Ca2+ currents, acting on cell surface channels.

Chemical Structure

GZ4

CAS#68312-88-9

Theoretical Analysis

MedKoo Cat#: 563086

Name: GZ4

CAS#: 68312-88-9

Chemical Formula: C11H17NO2

Exact Mass: 195.1259

Molecular Weight: 195.26

Elemental Analysis: C, 67.66; H, 8.78; N, 7.17; O, 16.39

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

GZ4; GZ-4; GZ 4;

IUPAC/Chemical Name

2-Aminoadamantane-1-carboxylic acid

InChi Key

KNDWUKJAYRIVHS-UHFFFAOYSA-N

InChi Code

InChI=1S/C11H17NO2/c12-9-8-2-6-1-7(3-8)5-11(9,4-6)10(13)14/h6-9H,1-5,12H2,(H,13,14)

SMILES Code

O=C(C12C(N)C3CC(C2)CC(C3)C1)O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 195.26 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Zoidis G, Sandoval A, Pineda-Farias JB, Granados-Soto V, Felix R. Anti-allodynic effect of 2-(aminomethyl)adamantane-1-carboxylic acid in a rat model of neuropathic pain: a mechanism dependent on CaV2.2 channel inhibition. Bioorg Med Chem. 2014 Mar 15;22(6):1797-803. doi: 10.1016/j.bmc.2014.02.006. Epub 2014 Feb 15. PubMed PMID: 24582401. 2: Xiao H, Liang W, Wang Y, Zhang J, Luo K. [Analysis of eleven isolated transfusion transmitted virus genotype]. Zhonghua Gan Zang Bing Za Zhi. 2001 Apr;9(2):89-91. Chinese. PubMed PMID: 11350686. 3: Auböck J, Niederwieser D, Romani N, Fritsch P, Huber C. Human interferon-gamma induces expression of HLA-DR on keratinocytes and melanocytes. Arch Dermatol Res. 1985;277(4):270-5. PubMed PMID: 3923947.