RS 100235 |CAS#171859-02-2 |5-HT4 Serotonin Receptor

MedKoo Cat#: 532580 | Name: RS 100235

Description:

WARNING: This product is for research use only, not for human or veterinary use.

RS 100235 is a 5-HT4 Serotonin Receptor.

Chemical Structure

RS 100235

CAS#171859-02-2

Theoretical Analysis

MedKoo Cat#: 532580

Name: RS 100235

CAS#: 171859-02-2

Chemical Formula: C27H35ClN2O5

Exact Mass: 502.2234

Molecular Weight: 503.04

Elemental Analysis: C, 64.47; H, 7.01; Cl, 7.05; N, 5.57; O, 15.90

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

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Related CAS #

No Data

Synonym

RS 100235; RS-100235; RS100235.

IUPAC/Chemical Name

1-(5-amino-6-chloro-2,3-dihydro-1,4-benzodioxin-8-yl)-3-[1-[3-(3,4-dimethoxyphenyl)propyl]piperidin-4-yl]propan-1-one

InChi Key

UVOCSZKGWJOKNN-UHFFFAOYSA-N

InChi Code

InChI=1S/C27H35ClN2O5/c1-32-23-8-6-19(16-24(23)33-2)4-3-11-30-12-9-18(10-13-30)5-7-22(31)20-17-21(28)25(29)27-26(20)34-14-15-35-27/h6,8,16-18H,3-5,7,9-15,29H2,1-2H3

SMILES Code

O=C(C1=C(OCCO2)C2=C(N)C(Cl)=C1)CCC3CCN(CCCC4=CC=C(OC)C(OC)=C4)CC3

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 503.04 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Chapple CR, Radley SC, Martin SW, Sellers DJ, Chess-Williams R. Serotonin-induced potentiation of cholinergic responses to electrical field stimulation in normal and neurogenic overactive human detrusor muscle. BJU Int. 2004 Mar;93(4):599-604. PubMed PMID: 15008739. 2: Sellers DJ, Chess-Williams R, Chapple CR. 5-Hydroxytryptamine-induced potentiation of cholinergic responses to electrical field stimulation in pig detrusor muscle. BJU Int. 2000 Oct;86(6):714-8. PubMed PMID: 11069383.