MedKoo Cat#: 531749 | Name: CP 94253 hydrochloride
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Description:

WARNING: This product is for research use only, not for human or veterinary use.

CP 94253 hydrochloride is a potent and selective serotonin 5-HT1B receptor agonist, with Ki values to be 2 nM for 5-HT1B and 89, 860, 49 and 1600 nM for 5-HT1A, 5-HT1C, 5-HT1D and 5-HT2 receptors respectively.

Chemical Structure

CP 94253 hydrochloride
CP 94253 hydrochloride
CAS#845861-39-4 (HCl)

Theoretical Analysis

MedKoo Cat#: 531749

Name: CP 94253 hydrochloride

CAS#: 845861-39-4 (HCl)

Chemical Formula: C15H20ClN3O

Exact Mass: 0.0000

Molecular Weight: 293.80

Elemental Analysis: C, 61.32; H, 6.86; Cl, 12.07; N, 14.30; O, 5.45

Price and Availability

Size Price Availability Quantity
10mg USD 350.00 2 Weeks
25mg USD 750.00 2 Weeks
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Synonym
CP 94253 hydrochloride; CP 94253 HCl; CP94253; CP-94253; CP 94253;
IUPAC/Chemical Name
5-propoxy-3-(1,2,3,6-tetrahydro-4-pyridinyl)-1H-pyrrolo[3,2-b]pyridine, monohydrochloride
InChi Key
PIIOXKQIZCVXMD-UHFFFAOYSA-N
InChi Code
InChI=1S/C15H19N3O.ClH/c1-2-9-19-14-4-3-13-15(18-14)12(10-17-13)11-5-7-16-8-6-11;/h3-5,10,16-17H,2,6-9H2,1H3;1H
SMILES Code
CCCOC1=CC=C(NC=C2C3=CCNCC3)C2=N1.[H]Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 293.80 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Najar F, Nasehi M, Haeri-Rohani SA, Zarrindast MR. The involvement of medial septum 5-HT1 and 5-HT2 receptors on ACPA-induced memory consolidation deficit: possible role of TRPC3, TRPC6 and TRPV2. J Psychopharmacol. 2015 Nov;29(11):1200-8. doi: 10.1177/0269881115609021. PubMed PMID: 26464456. 2: Nonogaki K, Kaji T. Pharmacological stimulation of serotonin 5-HT1B receptors enhances increases in plasma active glucagon-like peptide-1 levels induced by dipeptidyl peptidase-4 inhibition independently of feeding in mice. Diabetes Metab. 2015 Nov;41(5):425-8. doi: 10.1016/j.diabet.2015.06.005. PubMed PMID: 26234524.