CGP 55845 HCl is a potent, selective GABAB receptor antagonist (IC50 = 5 nM) that prevents agonist binding (pKi = 8.35) and inhibits GABA and glutamate release (pEC50 values are 8.08 and 7.85 respectively).
MedKoo Cat#: 513676
Name: CGP55845 HCl
CAS#: 149184-22-5 (HCl)
Chemical Formula: C18H23Cl3NO3P
Exact Mass: 0.0000
Molecular Weight: 438.70
Elemental Analysis: C, 49.28; H, 5.28; Cl, 24.24; N, 3.19; O, 10.94; P, 7.06
The following data is based on the product molecular weight 438.70 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
