Fenclonine acts as a selective and irreversible inhibitor of tryptophan hydroxylase, which is a rate-limiting enzyme in the biosynthesis of serotonin. It has been used experimentally to treat carcinoid syndrome.
MedKoo Cat#: 525042
Name: Fenclonine
CAS#: 7424-00-2
Chemical Formula: C9H10ClNO2
Exact Mass: 199.0400
Molecular Weight: 199.63
Elemental Analysis: C, 54.15; H, 5.05; Cl, 17.76; N, 7.02; O, 16.03
Solvent | mg/mL | mM | |
---|---|---|---|
Solubility | |||
DMSO | 1.5 | 7.51 | |
Water | 2.0 | 10.02 |
The following data is based on the product molecular weight 199.63 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |