CP-866087 | CAS#519052-02-9 | Mu-opioid Receptor Antagonist

MedKoo Cat#: 524876 | Name: CP-866087

Description:

WARNING: This product is for research use only, not for human or veterinary use.

CP-866087 is a selective mu-opioid receptor antagonist.

Chemical Structure

CP-866087

CAS#519052-02-9 (free base)

Theoretical Analysis

MedKoo Cat#: 524876

Name: CP-866087

CAS#: 519052-02-9 (free base)

Chemical Formula: C24H30N2O3S

Exact Mass: 426.1977

Molecular Weight: 426.57

Elemental Analysis: C, 67.58; H, 7.09; N, 6.57; O, 11.25; S, 7.52

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

519052-02-9 (free base) 519052-03-0 (mesylate)

Synonym

CP-866087; CP866087; CP 866087; UNII-MDH21334PI; CP-866,087.

IUPAC/Chemical Name

Methanesulfonamide, N-(3-(3-((2,3-dihydro-2-hydroxy-1H-inden-2-yl)methyl)-6-ethyl-3-azabicyclo(3.1.0)hex-6-yl)phenyl)-

InChi Key

ZBVPUFSKFGYNLC-FIDNPTQWSA-N

InChi Code

InChI=1S/C24H30N2O3S/c1-3-24(19-9-6-10-20(11-19)25-30(2,28)29)21-14-26(15-22(21)24)16-23(27)12-17-7-4-5-8-18(17)13-23/h4-11,21-22,25,27H,3,12-16H2,1-2H3/t21-,22+,24+

SMILES Code

CC[C@@]1([C@H]2[C@@H]1CN(C2)CC3(Cc4ccccc4C3)O)c5cccc(c5)NS(=O)(=O)C

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

Soluble in DMSO, not in water

Shelf Life

>2 years if stored properly

Drug Formulation

This drug may be formulated in DMSO

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 426.57 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Orri M, Abraham L, Giraldi A. A phase 2a multicenter, double-blind, placebo-controlled, crossover trial to investigate the efficacy, safety, and toleration of CP-866,087 (a high-affinity mu-opioid receptor antagonist) in premenopausal women diagnosed with female sexual arousal disorder (FSAD). J Sex Med. 2013 Oct;10(10):2484-96. doi: 10.1111/jsm.12071. Epub 2013 Jan 24. PubMed PMID: 23347610.