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MedKoo Cat#: 524648 | Name: Cgp 8065

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Cgp 8065 is a filaricidal compound, a dithiocarbamate-derivative of amoscanate.

Chemical Structure

Cgp 8065
Cgp 8065
CAS#62939-04-2

Theoretical Analysis

MedKoo Cat#: 524648

Name: Cgp 8065

CAS#: 62939-04-2

Chemical Formula: C16H15N3O4S2

Exact Mass: 377.0504

Molecular Weight: 377.44

Elemental Analysis: C, 50.91; H, 4.01; N, 11.13; O, 16.96; S, 16.99

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
Cgp 8065; Cgp8065; Cgp-8065.
IUPAC/Chemical Name
Propanoic acid, 3-((((4-((4-nitrophenyl)amino)phenyl)amino)thioxomethyl)thio)-
InChi Key
CTOSDJOWBFXFCP-UHFFFAOYSA-N
InChi Code
InChI=1S/C16H15N3O4S2/c20-15(21)9-10-25-16(24)18-13-3-1-11(2-4-13)17-12-5-7-14(8-6-12)19(22)23/h1-8,17H,9-10H2,(H,18,24)(H,20,21)
SMILES Code
C(CCSC(=S)Nc1ccc(cc1)Nc1ccc(cc1)[N+](=O)[O-])(=O)O
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 377.44 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Walter RD, Kuhlow F. Parasite-specific interaction of N-[4-(4'nitroanilino)-phenyl]-S-(beta-carboxyethyl)-dithiocar bamic acid-ester with arginyl-tRNA-synthetase from Dirofilaria immitis. Trop Med Parasitol. 1985 Dec;36(4):230-2. PubMed PMID: 3841408. 2: Walter RD, Albiez E. Parasite-specific inhibition of 5'-nucleotidase from Onchocerca volvulus and Dirofilaria immitis by the amoscanate-derivative CGP 8065. Mol Biochem Parasitol. 1985 Aug;16(2):109-15. PubMed PMID: 2993882. 3: Walter RD, Ossikovski E. Effect of amoscanate derivative CGP 8065 on aminoacyl-tRNA synthetases in Ascaris suum. Mol Biochem Parasitol. 1985 Jan;14(1):23-8. PubMed PMID: 3838573.

View History

CGP-20712

CGP-20712