OUP-16 is a potent and selective histamine H4 receptor agonist. OUP-16 is a full hH4R agonist with 40-fold selectivity over the hH3R and superior to its (2S,5S)-configured optical antipode. The H4R is expressed in various cells of the immune system, suggesting a role in inflammatory, autoimmune, and allergic disorders.
MedKoo Cat#: 522692
Name: OUP-16
CAS#: 1038917-11-1
Chemical Formula: C11H16N6O
Exact Mass: 248.1386
Molecular Weight: 248.29
Elemental Analysis: C, 53.21; H, 6.50; N, 33.85; O, 6.44
The following data is based on the product molecular weight 248.29 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
