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MedKoo Cat#: 319814 | Name: Revamilast

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Revamilast, also known as GRC4039, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritis

Chemical Structure

Revamilast
Revamilast
CAS#893555-90-3 (free)

Theoretical Analysis

MedKoo Cat#: 319814

Name: Revamilast

CAS#: 893555-90-3 (free)

Chemical Formula: C18H9Cl2F2N3O4

Exact Mass: 438.9938

Molecular Weight: 440.18

Elemental Analysis: C, 49.12; H, 2.06; Cl, 16.11; F, 8.63; N, 9.55; O, 14.54

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
893555-91-4 (sodium) 893555-90-3 (free) 1026382-18-2 (tautomer)
Synonym
GRC4039; GRC-4039; GRC 4039; Revamilast
IUPAC/Chemical Name
3,5-Dichloro-4-((6-(difluoromethoxy)(1)benzofuro(3,2-c)pyridine-9-yl)carboxamido)pyridine 1-oxide
InChi Key
IXQHNBONEVULTL-UHFFFAOYSA-N
InChi Code
InChI=1S/C18H9Cl2F2N3O4/c19-10-6-25(27)7-11(20)15(10)24-17(26)8-1-2-13(29-18(21)22)16-14(8)9-5-23-4-3-12(9)28-16/h1-7,18H,(H,24,26)
SMILES Code
O=C(C1=CC=C(OC(F)F)C(O2)=C1C3=C2C=CN=C3)NC4=C(Cl)C=[N+]([O-])C=C4Cl
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
Soluble in DMSO, not in water
Shelf Life
>2 years if stored properly
Drug Formulation
This drug may be formulated in DMSO
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 440.18 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL

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