Pravadoline, also known as WIN 48098-6, is a agonist of the cannabinoid receptor. Pravadoline inhibited the synthesis of prostaglandins (PGs) in mouse brain both in vitro (IC50, 4.9 microM) and ex vivo (ED50, 20 mg/kg p.o.) and displayed antinociceptive activity in rodents subjected to a variety of chemical, thermal and mechanical nociceptive stimuli.
MedKoo Cat#: 127549
Name: Pravadoline maleate
CAS#: 92623-84-2 (maleate)
Chemical Formula: C27H30N2O7
Exact Mass: 494.2053
Molecular Weight: 494.54
Elemental Analysis: C, 65.57; H, 6.11; N, 5.66; O, 22.65
The following data is based on the product molecular weight 494.54 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
50 mM | 0.02 mL | 0.12 mL | 0.23 mL |