MedKoo Cat#: 127402 | Name: Tipindole

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Tipindole is serotonin antagonist. It is also a monamine oxidase inhibitor. Tipindole exerts no effect on the serotonin-induced contraction and relaxation of the bladder detrusor. Tipindole depresses reflexes from pericardial receptors considerably more than reflexes from carotid sinus receptors.

Chemical Structure

Tipindole
CAS#7489-66-9

Theoretical Analysis

MedKoo Cat#: 127402

Name: Tipindole

CAS#: 7489-66-9

Chemical Formula: C16H20N2O2S

Exact Mass: 304.1245

Molecular Weight: 304.41

Elemental Analysis: C, 63.13; H, 6.62; N, 9.20; O, 10.51; S, 10.53

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
No Data
Synonym
TIPINDOLE; tipindole [INN]
IUPAC/Chemical Name
2-(dimethylamino)ethyl 1,3,4,5-tetrahydrothiopyrano[4,3-b]indole-8-carboxylate
InChi Key
WNDHLINIYZAWCR-UHFFFAOYSA-N
InChi Code
InChI=1S/C16H20N2O2S/c1-18(2)6-7-20-16(19)11-3-4-14-12(9-11)13-10-21-8-5-15(13)17-14/h3-4,9,17H,5-8,10H2,1-2H3
SMILES Code
CN(C)CCOC(=O)C1=CC2=C(NC3=C2CSCC3)C=C1
Appearance
To be determined
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 -4 C for short term (days to weeks) or -20 C for long term(months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 304.41 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1: Demina LM, Zbarskaia IS, Pidevich IN. Farmakologicheskiĭ analiz mekhanizma vozniknoveniia serotoninovoĭ diarei u mysheĭ [Pharmacologic analysis of the mechanism of development of serotonin diarrhea in the mouse]. Farmakol Toksikol. 1981 Jan-Feb;44(1):91-2. Russian. PMID: 7262307.