CDK12-IN-5, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 23.9 nM at high ATP (2 mM).
MedKoo Cat#: 126613
Name: CDK12-IN-5
CAS#: 2651200-35-8
Chemical Formula: C18H15F5N8O
Exact Mass: 454.1289
Molecular Weight: 454.37
Elemental Analysis: C, 47.58; H, 3.33; F, 20.91; N, 24.66; O, 3.52
The following data is based on the product molecular weight 454.37 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
