Enerisant is a histamine H3 receptor antagonist. In H3 receptor binding assay using (R)-α-methyl[3H]histamine, Enerisant showed IC50 of 4.9 nM. Enerisant may be useful for the treatment of Alzheimer's disease, schizophrenia, etc.
MedKoo Cat#: 125459
Name: Enerisant hydrochloride dihydrate
CAS#: 1152749-09-1 (HCl 2H2O)
Chemical Formula: C22H35ClN4O5
Exact Mass: 470.2300
Molecular Weight: 471.00
Elemental Analysis: C, 56.10; H, 7.49; Cl, 7.53; N, 11.90; O, 16.98
The following data is based on the product molecular weight 471.00 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
