MedKoo Biosciences, Inc.
Tel:   +1-919-636-5577    Fax:   +1-919-980-4831    Email:   sales@medkoo.com
Search
Login Register
Search
MedKoo Cat#: 124825 | Name: Buntanetap tartrate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Buntanetap, also known as R-phenserine or (-)-Phenserine, is a selective, non-competitive inhibitor of acetylcholinesterase (AChE). (-)-Phenserine produces rapid, potent, and long-lasting AChE inhibition, in vivo. (-)-Phenserine attenuates soman-induced neuropathology.

Chemical Structure

Buntanetap tartrate
Buntanetap tartrate
CAS#865795-23-9 (racemic tartrate)

Theoretical Analysis

MedKoo Cat#: 124825

Name: Buntanetap tartrate

CAS#: 865795-23-9 (racemic tartrate)

Chemical Formula: C24H29N3O8

Exact Mass: 487.2000

Molecular Weight: 487.51

Elemental Analysis: C, 59.13; H, 6.00; N, 8.62; O, 26.25

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
Bulk Inquiry
Related CAS #
101246-66-6 (free base) 156910-61-1 (tartrate) 159652-53-6 (racemic) 865795-23-9 (tartrate)
Synonym
Posiphen tartrate; Buntanetap tartrate; R-Phenserine tartrate; G18HAS9LKM
IUPAC/Chemical Name
(3aR,8aS)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-yl phenylcarbamate (2R,3R)-2,3-dihydroxysuccinate
InChi Key
XKKPTCVQEJZDGT-UHFFFAOYSA-N
InChi Code
InChI=1S/C20H23N3O2.C4H6O6/c1-20-11-12-22(2)18(20)23(3)17-10-9-15(13-16(17)20)25-19(24)21-14-7-5-4-6-8-14;5-1(3(7)8)2(6)4(9)10/h4-10,13,18H,11-12H2,1-3H3,(H,21,24);1-2,5-6H,(H,7,8)(H,9,10)
SMILES Code
O[C@H]([C@@H](O)C(O)=O)C(O)=O.[H][C@@]12N(C)CC[C@]1(C)C3=C(C=CC(OC(=O)NC4=CC=CC=C4)=C3)N2C
Appearance
To be determined
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 487.51 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
Vofo BN, Chowers I. Suppressing Inflammation for the Treatment of Diabetic Retinopathy and Age-Related Macular Degeneration: Dazdotuftide as a Potential New Multitarget Therapeutic Candidate. Biomedicines. 2023 May 27;11(6):1562. doi: 10.3390/biomedicines11061562. PMID: 37371657; PMCID: PMC10295757.