M4205, also known as IDRX-42, is A Highly Selective Inhibitor of KIT Mutations for Treatment of Unresectable Metastatic or Recurrent Gastrointestinal Stromal Tumors. M4205 has a superior profile compared to approved drugs, suggesting a best-in-class potential for recurrent and metastatic GISTs driven by KIT mutations.
MedKoo Cat#: 122722
Name: M4205
CAS#: 2590556-80-0
Chemical Formula: C29H32N8O
Exact Mass: 508.2699
Molecular Weight: 508.63
Elemental Analysis: C, 68.48; H, 6.34; N, 22.03; O, 3.15
The following data is based on the product molecular weight 508.63 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 1 mM | 1.15 mL | 5.76 mL | 11.51 mL |
| 5 mM | 0.23 mL | 1.15 mL | 2.3 mL |
| 10 mM | 0.12 mL | 0.58 mL | 1.15 mL |
| 50 mM | 0.02 mL | 0.12 mL | 0.23 mL |
