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MedKoo Cat#: 577727 | Name: Azilsartan mepixetil

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Azilsartan mepixetil is an angiotensin II receptor antagonist with renal and cardioprotective effects.

Chemical Structure

Azilsartan mepixetil
Azilsartan mepixetil
CAS#1596357-16-2 (free base)

Theoretical Analysis

MedKoo Cat#: 577727

Name: Azilsartan mepixetil

CAS#: 1596357-16-2 (free base)

Chemical Formula: C36H34N6O8

Exact Mass: 678.2438

Molecular Weight: 678.70

Elemental Analysis: C, 63.71; H, 5.05; N, 12.38; O, 18.86

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.
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Related CAS #
1596357-16-2 (free base) 2153458-32-1 (potassium)
Synonym
Azilsartan mepixetil
IUPAC/Chemical Name
rac-(1R)-1-({[(3,5,6-trimethylpyrazin-2-yl)methoxy]carbonyl}oxy)ethyl 2-ethoxy-1-{[2'-(5-oxo-2,5-dihydro-1,2,4-oxadiazol-3-yl)[1,1'-biphenyl]-4-yl]methyl}-1H-benzimidazole-7-carboxylate
InChi Key
JXSDNNVNQNYJSP-HSZRJFAPSA-N
InChi Code
InChI=1S/C36H34N6O8/c1-6-46-34-39-29-13-9-12-28(33(43)48-23(5)49-36(45)47-19-30-22(4)37-20(2)21(3)38-30)31(29)42(34)18-24-14-16-25(17-15-24)26-10-7-8-11-27(26)32-40-35(44)50-41-32/h7-17,23H,6,18-19H2,1-5H3,(H,40,41,44)/t23-/m1/s1
SMILES Code
O=C(C1=C2C(N=C(OCC)N2CC3=CC=C(C4=CC=CC=C4C5=NC(ON5)=O)C=C3)=CC=C1)O[C@H](OC(OCC6=NC(C)=C(C)N=C6C)=O)C
Appearance
Solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition
Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility
To be determined
Shelf Life
>2 years if stored properly
Drug Formulation
To be determined
Stock Solution Storage
0 - 4 C for short term (days to weeks), or -20 C for long term (months).
HS Tariff Code
2934.99.9001
More Info

Preparing Stock Solutions

The following data is based on the product molecular weight 678.70 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Recalculate based on batch purity %
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.15 mL 5.76 mL 11.51 mL
5 mM 0.23 mL 1.15 mL 2.3 mL
10 mM 0.12 mL 0.58 mL 1.15 mL
50 mM 0.02 mL 0.12 mL 0.23 mL
1. Hardin MD, Jacobs TF. Azilsartan. 2021 Jul 19. In: StatPearls [Internet]. Treasure Island (FL): StatPearls Publishing; 2022 Jan–. PMID: 30860708. 2. Lam S. Azilsartan: a newly approved angiotensin II receptor blocker. Cardiol Rev. 2011 Nov-Dec;19(6):300-4. doi: 10.1097/CRD.0b013e31822e9ba3. PMID: 21983318.