CHIR98024 | CAS#

MedKoo Cat#: 556003 | Name: CHIR98024

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Description:

WARNING: This product is for research use only, not for human or veterinary use.

CHIR98024, also known as CT-98024, is a potent GSK3 Inhibitor with IC50=1 nM. CHIR98024 is an isomer of CHIR98014, both of which structure are very similar. Many vendors confused each other.

Chemical Structure

CHIR98024

CAS#556813-39-9 (CHIR98024)

Theoretical Analysis

MedKoo Cat#: 556003

Name: CHIR98024

CAS#: 556813-39-9 (CHIR98024)

Chemical Formula: C20H17Cl2N9O2

Exact Mass: 485.0882

Molecular Weight: 486.32

Elemental Analysis: C, 49.40; H, 3.52; Cl, 14.58; N, 25.92; O, 6.58

Price and Availability

Size	Price	Availability	Quantity
10mg	USD 400.00	2 Weeks
25mg	USD 850.00	2 Weeks

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Related CAS #

556813-39-9 (CHIR98024) 252935-94-7 (CHIR98014) CHIR98014 HCl

Synonym

CHIR98024; CHIR-98024; CHIR 98024; CT-98024; CT 98024; CT98024; CHIR98014-isomer; CHIR-98014-isomer; CHIR 98014-isomer; CT-98014-isomer; CT 98014-isomer; CT98014-isomer;

IUPAC/Chemical Name

N6-[2-[[4-(2,4-Dichlorophenyl)-5-(1H-imidazol-2-yl)-2-pyrimidinyl]amino]ethyl]-3-nitro-2,6-pyridinediamine

InChi Key

NDFXSHIIGXVOKT-UHFFFAOYSA-N

InChi Code

InChI=1S/C20H17Cl2N9O2/c21-11-1-2-12(14(22)9-11)17-13(19-25-6-7-26-19)10-28-20(30-17)27-8-5-24-16-4-3-15(31(32)33)18(23)29-16/h1-4,6-7,9-10H,5,8H2,(H,25,26)(H3,23,24,29)(H,27,28,30)

SMILES Code

NC1=NC(NCCNC2=NC=C(C3=NC=CN3)C(C4=CC=C(Cl)C=C4Cl)=N2)=CC=C1[N+]([O-])=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 486.32 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

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