Endralazine mesylate | CAS# 65322-72-7 | Antihypertensive

MedKoo Cat#: 414012 | Name: Endralazine mesylate

Description:

WARNING: This product is for research use only, not for human or veterinary use.

Endralazine mesylate is an Antihypertensive

Chemical Structure

Endralazine mesylate

CAS#65322-72-7

Theoretical Analysis

MedKoo Cat#: 414012

Name: Endralazine mesylate

CAS#: 65322-72-7

Chemical Formula: C15H19N5O4S

Exact Mass: 365.1158

Molecular Weight: 365.41

Elemental Analysis: C, 49.31; H, 5.24; N, 19.17; O, 17.51; S, 8.77

Price and Availability

This product is currently not in stock but may be available through custom synthesis. To ensure cost efficiency, the minimum order quantity is 1 gram. The estimated lead time is 2 to 4 months, with pricing dependent on the complexity of the synthesis (typically high for intricate chemistries). Quotes for quantities below 1 gram will not be provided. To request a quote, please click the button below. Note: If this product becomes available in stock in the future, pricing will be listed accordingly.

Bulk Inquiry

Related CAS #

No Data

Synonym

Endralazine mesylate; NSC310289; NSC-310289; NSC 310289

IUPAC/Chemical Name

Pyrido(4,3-c)pyridazin-3(2H)-one, 6-benzoyl-5,6,7,8-tetrahydro-, hydrazone, monomethanesulfonate

InChi Key

HMVROCAATOPFHB-UHFFFAOYSA-N

InChi Code

InChI=1S/C14H15N5O.CH4O3S/c15-16-13-8-11-9-19(7-6-12(11)17-18-13)14(20)10-4-2-1-3-5-10;1-5(2,3)4/h1-5,8H,6-7,9,15H2,(H,16,18);1H3,(H,2,3,4)

SMILES Code

O=C(N(C1)CCC(C1=C/2)=NNC2=N/N)C3=CC=CC=C3.CS(=O)(O)=O

Appearance

Solid powder

Purity

>98% (or refer to the Certificate of Analysis)

Shipping Condition

Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Storage Condition

Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

Solubility

To be determined

Shelf Life

>2 years if stored properly

Drug Formulation

To be determined

Stock Solution Storage

0 - 4 C for short term (days to weeks), or -20 C for long term (months).

HS Tariff Code

2934.99.9001

More Info

Instruction

View handling instruction

Preparing Stock Solutions

The following data is based on the product molecular weight 365.41 Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.15 mL	5.76 mL	11.51 mL
5 mM	0.23 mL	1.15 mL	2.3 mL
10 mM	0.12 mL	0.58 mL	1.15 mL
50 mM	0.02 mL	0.12 mL	0.23 mL

1: Kindler J, Mödder G, Sieberth HG. Autoradiographische Untersuchungen zur Verteilung von 14C-Endralazin bei der Maus [Autoradiographic studies of the distribution of 14C-endralazine in the mouse]. Arzneimittelforschung. 1985;35(3):599-602. German. PMID: 4039585. 2: Bechter R, Schön H. Use of the whole-embryo culture system in drug safety assessment? Toxicol In Vitro. 1988;2(3):195-203. doi: 10.1016/0887-2333(88)90008-2. PMID: 20702335.